Methyltestosterone for Sale – Potent Oral Androgen for Rapid Performance Enhancement
Methyltestosterone: One of the Oldest Oral Testosterone Derivatives
What Is Methyltestosterone?
Methyltestosterone is a synthetic oral form of testosterone, modified for oral bioavailability by the addition of a methyl group at the 17-alpha position. This alteration allows it to survive first-pass liver metabolism, making it effective when taken by mouth. It was one of the earliest anabolic steroids developed (1930s) and has been used medically for male hypogonadism, delayed puberty, and menopausal symptoms in women.
Chemical & Pharmacological Profile
Chemical Name: 17α-methyltestosterone
Brand Names: Android, Testred, Virilon
Form: Oral tablet (occasionally sublingual)
Half-Life: ~3–4 hours
Class: Androgen; Anabolic steroid
Liver Toxicity: High (17α-alkylated)
Anabolic:Androgenic Ratio: Moderate anabolic, highly androgenic
Key Effects and Benefits
Quick Elevation of Testosterone: Raises testosterone levels rapidly — often used short-term for testosterone boosts.
Increased Strength and Aggression: Provides notable androgenic stimulation, often boosting mental drive and intensity.
Medical Use in Hormone Therapy: Still prescribed in some cases for low testosterone, delayed puberty, or menopausal support (in women).
Rare in Bodybuilding Today: Due to side effects, it's mostly replaced by safer and more effective alternatives.
Typical Dosage
| Use Case | Dosage Range | Duration |
|---|---|---|
| Men (TRT/Performance) | 10–40 mg/day | 2–4 weeks |
| Women (medical use) | 2.5–10 mg/day | Short-term only |
| Bodybuilding (rare) | 20–50 mg/day | 2–4 weeks |
Use beyond short cycles is not recommended due to liver strain and androgenic side effects.
Side Effects
Methyltestosterone is considered harsh due to its high androgenic activity and liver toxicity:
Common Side Effects
Liver Toxicity: Strongly hepatotoxic—can elevate liver enzymes and risk of liver damage
Estrogenic Effects: Aromatizes into estrogen → gynecomastia, water retention, bloating
Androgenic Effects: Acne, hair loss, oily skin, body hair growth
Mood Swings & Aggression: Strong psychological effects in some users
Testosterone Suppression: Shuts down natural testosterone production → requires PCT
Summary: Is Methyltestosterone Worth Using?
Methyltestosterone is a historically important steroid that offers fast testosterone elevation and androgenic benefits. However, it's largely considered outdated and harsh due to its high toxicity, estrogenic activity, and limited anabolic benefits compared to safer compounds like Testosterone Propionate, Anavar, or Turinabol.
Best suited for:
Short-term testosterone support in clinical settings
Occasional use in aggression or strength-based sports (with caution)
Not recommended for:
Long-term performance enhancement
Women (due to virilization risk)
Liver-sensitive users or beginners
